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Clinical Efficacy and Target Engagement of Glutamatergic Drugs: Placebo-Controlled RCTs of Pomaglumetad and TS-134 for Reversal of Ketamine-Induced Psychotic Symptoms and PharmacoBOLD in Healthy Volunteers

2020-03-12 psychiatry and clinical psychology Title + abstract only
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We tested two metabotropic glutamate receptor 2/3 (mGluR2/3) agonist prodrugs - pomaglumetad (POMA) and TS-134 - including a high-dose of POMA that was four times the dose tested in the failed phase schizophrenia III trials - in two proof of mechanism, Phase Ib studies using identical pharmacoBOLD target-engagement methodology. The POMA study was a double-blind, NIMH-sponsored, 10-day study of 80 or 320 mg/d POMA or placebo (1:1:1 ratio), designed to detect d>0.8 sd between-group effect-size di...

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